Thoas Fioretos
Research team manager
Interleukin 4 induces apoptosis of acute myeloid leukemia cells in a Stat6 dependent manner
Author
Summary, in English
Cytokines provide signals that regulate immature normal and acute myeloid leukemia (AML) cells in the bone marrow microenvironment. We here identify interleukin 4 (IL4) as a selective inhibitor of AML cell growth and survival in a cytokine screen using fluorescently labeled AML cells. RNA-sequencing of the AML cells revealed an IL4-induced upregulation of Stat6 target genes and enrichment of apoptosis-related gene expression signatures. Consistent with these findings, we found that IL4 stimulation of AML cells induced Stat6 phosphorylation and that disruption of Stat6 using CRISPR/Cas9-genetic engineering rendered cells partially resistant to IL4-induced apoptosis. To evaluate whether IL4 inhibits AML cells in vivo, we expressed IL4 ectopically in AML cells transplanted into mice and also injected IL4 into leukemic mice; both strategies resulted in the suppression of the leukemia cell burden and increased survival. Notably, IL4 exposure caused reduced growth and survival of primary AML CD34(+)CD38(-) patient cells from several genetic subtypes of AML, whereas normal stem and progenitor cells were less affected. The IL4-induced apoptosis of AML cells was linked to Caspase-3 activation. Our results demonstrate that IL4 selectively induces apoptosis of AML cells in a Stat6-dependent manner, findings that may translate into new therapeutic opportunities in AML.Leukemia accepted article preview online, 18 August 2017. doi:10.1038/leu.2017.261.
Department/s
- Division of Clinical Genetics
- Translational Genomic and Functional Studies of Leukemia
- Division of Molecular Medicine and Gene Therapy
- BioCARE: Biomarkers in Cancer Medicine improving Health Care, Education and Innovation
- StemTherapy: National Initiative on Stem Cells for Regenerative Therapy
Publishing year
2018
Language
English
Pages
588-596
Publication/Series
Leukemia
Volume
32
Issue
3
Document type
Journal article
Publisher
Nature Publishing Group
Topic
- Cell and Molecular Biology
Keywords
- Journal Article
Status
Published
Project
- Identification and characterization of candidate therapeutic targets in acute myeloid leukemia
Research group
- Translational Genomic and Functional Studies of Leukemia
ISBN/ISSN/Other
- ISSN: 1476-5551